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Table 2 Drugs in the minimal hitting sets

From: Optimal drug combinations and minimal hitting sets

NSC

Name

Mechanism of action

21206

6-aminonicotinamide

Antimetabolite

174121

methotrexate derivative

Antimetabolite

606698

Rapamycin prodrug

mTOR inhibitor

606699

Rapamycin prodrug

mTOR inhibitor

147340

Anisomycin hydrochloride

NA

646846

bengamide B

NA

656238

2-Methyl-4,8-dihydrobenzo [1,2-b:5,4-b']dithiophene-4,8-dione

NA

656240

2-Hydroxymethyl-4,8-dihydrobenzo [1,2-b:5,4-b']dithiophene-4,8-dione

NA

671526

Toxin.delta.53L

NA

674092

Quinoline-4-carboxamide, N, N'-[(1,4-piperazinediyl) bis(3,1-propanediyl)]bis(2-phenyl-, dihydrochloride

NA

676495

NA

NA

689535

1-methyl-3-(1-pyrazin-2-ylethylideneamino)-1-(2-pyridin-2-ylethyl) thiourea

NA

692745

1H-Inden-1-one, 2,3-dihydro-2-[(4-hydroxy-3,5-dimethylphenyl) methylene]-5,6-dimethoxy-, (2E)-

NA

623794

1,4-Benzodioxin-2-carboxamide, 6-(4-oxo-4-H-1-benzopyran-2-yl)-N-(3-pyridinylmethyl)-

NA

682449

Benzo [1,2-b:4,5-b']dithiophene-4,8-dione, 2-(1-hydroxyethyl)-

NA

691039

(7S)-7-hydroxy-1,2,3-trimethoxy-10-methylsulfanyl-6,7-dihydro-5H-benzo [a]heptalen-9-one

NA

725983

7-methoxy-5-oxo-8-[3-(9-oxo-9,10-dihydro-4-acridinylcarboxam ido)propoxyl]-(11aS)-1H,2H,3H,5H-bezo [e]pyrrolo [1,2-a][1,4]d iazepine

NA

  1. The list of drugs in the minimal hitting sets reported in Table 1. NSC stands for cancer chemotherapy National Service Center number. NA stands for Not Available.