Name | Description | Value | Units | Reference |
---|---|---|---|---|
K D, ATP | ATP-p38 affinity | 67 | uM | In-house measurement |
K D, ATF2 | ATF2-p38 affinity | 38 | uM | [30] |
K D, MK2 | MK2-p38 affinity | 20 | nM | [31] |
k cat, ATF2 | p38-ATF2 catalytic rate | 1.2 | s-1 | [30] |
k cat, MK2 | p38-MK2 catalytic rate | 0.17 2.4 | s-1 s-1 | [31] In-house measurement |
[p38] | p38 (active) initial condition | 0.5 | nM | Â |
[ATP] | ATP initial condition | 50 | uM | Â |
[ATF2] | ATF2 initial condition | 100 | nM | Â |
[MK2] | MK2 initial condition | 10 | nM | Â |